Omadacycline
Omadacycline
Definition
An aminomethylcycline and a semisynthetic tetracycline derivative, with antimicrobial activity. Upon administration, omadacycline binds to the bacterial 30S ribosomal subunit and inhibits bacterial protein synthesis. Omadacycline is engineered to overcome certain tetracycline resistance mechanisms, including tetracycline-specific efflux pumps and ribosomal protection.
Also known as (4S,4aS,5aR,12aS)-4,7-bis(dimethylamino)-9-{[(2,2-dimethylpropyl)amino]methyl}- 3,10,12,12a-tetrahydroxy-1,11-dioxo-1,4,4a,5,5a,6,11,12a-octahydrotetracene-2- carboxamide, 2-naphthacenecarboxamide, 4,7-bis(dimethylamino)-9-(((2,2-dimethylpropyl)amino)methyl)-1,4,4a,5,5a,6,11,12a-octahydro-3,10,12,12a-tetrahydroxy-1,11-dioxo-, (4s,4aS,5aR,12aS)-, 4-methylbenzenesulfonate (1:1), Amadacyclin, OMADACYCLINE, PTK 0796 — per NCIT
Also identified as
- ATC J01AA15 per RXNORM
- NCIT NCIT:C90688 per NCIT
- SCTID 781644002 per RXNORM
- SCTID 781654003 per RXNORM
- UNII 090IP5RV8F per RXNORM
Indications
| Disease | Relation | Source |
|---|---|---|
| Bacterial infectious disease | may prevent | MEDRT · Public domain (U.S. Government work) |
| Bacterial infectious disease | may treat | MEDRT · Public domain (U.S. Government work) |
| Bacterial pneumonia | may treat | MEDRT · Public domain (U.S. Government work) |
| Skin disease caused by bacterial infection | may treat | MEDRT · Public domain (U.S. Government work) |
Organ Effects
| Organ | Side effect / interaction | Source |
|---|---|---|
| Lungs | may treat a disease of this organ | DERIVED · CC BY 4.0 |
| Respiratory system | may treat a disease of this organ | DERIVED · CC BY 4.0 |
2 entries above are marked DERIVED: Atlas Médico inferred them by combining two sourced claims, and no source asserts these links directly. Treat them as a navigation aid, not as a clinical statement.