Ublituximab
Ublituximab
Definition
A chimeric recombinant IgG1 monoclonal antibody directed against human CD20 with potential antineoplastic activity. Ublituximab specifically binds to the B cell-specific cell surface antigen CD20, thereby potentially inducing a B cell-directed complement dependent cytotoxicity (CDC) and antibody-dependent cell-mediated cytotoxicity (ADCC) against CD20-expressing B cells, leading to B cell apoptosis. CD20 is a non-glycosylated cell surface phosphoprotein that is exclusively expressed on B cells during most stages of B cell development and is often overexpressed in B-cell malignancies. Ublituximab has a specific glycosylation profile, with a low fucose content, that may enhance its ADCC response against malignant B cells.
Also known as Briumvi, LFB R603, LFB-R603, LFBR603, TG 1101, TG 20, TG-1101, TG-20, TG1101, TG20, TGTX 1101, TGTX-1101, TGTX1101, UBLITUXIMAB, Ublituximab-xiiy — per NCIT
Also identified as
- ATC L04AG14 per RXNORM
- NCIT NCIT:C91078 per NCIT
- SCTID 1351582007 per RXNORM
- UNII U59UGK3IPC per RXNORM
Indications
| Disease | Relation | Source |
|---|---|---|
| Chronic progressive multiple sclerosis | may treat | MEDRT · Public domain (U.S. Government work) |
| Demyelinating disease | may treat | MEDRT · Public domain (U.S. Government work) |
| Relapsing-remitting multiple sclerosis | may treat | MEDRT · Public domain (U.S. Government work) |
Organ Effects
| Organ | Side effect / interaction | Source |
|---|---|---|
| Central nervous system | may treat a disease of this organ | DERIVED · CC BY 4.0 |
| Nervous system | may treat a disease of this organ | DERIVED · CC BY 4.0 |
2 entries above are marked DERIVED: Atlas Médico inferred them by combining two sourced claims, and no source asserts these links directly. Treat them as a navigation aid, not as a clinical statement.