Quinine

ATC Code P01BC01

Quinine

Definition

A quinidine alkaloid isolated from the bark of the cinchona tree. Quinine has many mechanisms of action, including reduction of oxygen intake and carbohydrate metabolism; disruption of DNA replication and transcription via DNA intercalation; and reduction of the excitability of muscle fibers via alteration of calcium distribution. This agent also inhibits the drug efflux pump P-glycoprotein which is overexpressed in multi-drug resistant tumors and may improve the efficacy of some antineoplastic agents. (NCI04)

Also known as (-)-Quinine, QUIN, QUININE — per NCIT

Also identified as

Indications

Disease Relation Source
Babesiosis may treat MEDRT · Public domain (U.S. Government work)
Plasmodium falciparum malaria may treat MEDRT · Public domain (U.S. Government work)