Dutasteride
Dutasteride
Definition
A synthetic 4-azasteroid compound. Dutasteride competitively and specifically binds to isoenzymes 1 and 2 of 5 alpha-reductase, forming stable enzyme complexes and inhibiting the conversion of testosterone to 5 alpha-dihydrotestosterone (DHT); the reduction in DHT activity may mitigate or prevent enlargement of the prostate gland. The type 2 5 alpha-reductase isoenzyme is primarily active in the reproductive tissues, while the type 1 isoenzyme is also active in skin and the liver.
Also known as alpha,alpha,alpha,alpha',alpha',alpha'-Hexafluoro-3-oxo-4-aza-5alpha-androst-1-ene-17beta-carboxy-2',5'-xylidide, Avodart, Avolve,(5alpha,17beta)-N-(2,5-Bis(trifluoromethyl)phenyl)-3-oxo-4-azaandrost-1-ene-17-carboxamide, DUTASTERIDE, GG 745, GG745 — per NCIT
Also identified as
- ATC G04CB02 per RXNORM
- NCIT NCIT:C47503 per NCIT
- SCTID 385570006 per RXNORM
- SCTID 385572003 per RXNORM
- UNII O0J6XJN02I per RXNORM
Indications
| Disease | Relation | Source |
|---|---|---|
| Benign prostatic hyperplasia | may treat | MEDRT · Public domain (U.S. Government work) |
Organ Effects
| Organ | Side effect / interaction | Source |
|---|---|---|
| Genitourinary system | may treat a disease of this organ | DERIVED · CC BY 4.0 |
| Male reproductive system | may treat a disease of this organ | DERIVED · CC BY 4.0 |
| Prostate | may treat a disease of this organ | DERIVED · CC BY 4.0 |
| Reproductive system | may treat a disease of this organ | DERIVED · CC BY 4.0 |
4 entries above are marked DERIVED: Atlas Médico inferred them by combining two sourced claims, and no source asserts these links directly. Treat them as a navigation aid, not as a clinical statement.