Eplerenone

ATC Code C03DA04

Eplerenone

Definition

A selective aldosterone receptor antagonist. Eplerenone binds to the mineralocorticoid receptor and blocks the binding of aldosterone, thereby decreasing sodium resorption and subsequently increasing water outflow. This leads to a decrease in blood pressure. Eplerenone is used in the treatment of hypertension and congestive heart failure.

Also known as 9,11alpha-Epoxy-17-hydroxy-3-oxo-17alpha-pregn-4-ene-7alpha,21-dicarboxylic acid, gamma-lactone, Methyl Ester, EPLERENONE, Inspra — per NCIT

Also identified as

Indications

Disease Relation Source
Hypertensive disorder may treat MEDRT · Public domain (U.S. Government work)
Systolic heart failure may treat MEDRT · Public domain (U.S. Government work)