Degarelix

ATC Code L02BX02

Degarelix

Definition

A long-acting, synthetic peptide with gonadotrophin-releasing hormone (GnRH) antagonistic properties. Degarelix targets and blocks GnRH receptors located on the surfaces of gonadotroph cells in the anterior pituitary, thereby reducing secretion of luteinizing hormone (LH) by pituitary gonadotroph cells and so decreasing testosterone production by interstitial (Leydig) cells in the testes.

Also known as ASP 3550, ASP-3550, ASP3550, DEGARELIX, FE 200486, FE-200486, FE200486, Firmagon — per NCIT

Also identified as

Indications

Disease Relation Source
Prostate cancer may treat MEDRT · Public domain (U.S. Government work)